产品编号:U821925
产品规格:500mg
产品价格:面议
| 标准品编号: | U821925 |
| 名称: | URB602 |
| 别名: | Biphenyl-3-yl Carbamic Acid, Cyclohexyl Ester; N-[1,1'-Biphenyl]-3-yl-carbamic Acid Cyclohexyl Ester |
| CAS号: | 565460-15-3 |
| 分子式: | C₁₉H₂₁NO₂ |
| 外观: | 白色固体 |
| 熔点: | 122-123°C |
| 分子量: | 295.38 |
| 溶解度: | DMSO |
| 类别: | Research Tools; Molecular Biology; Enzyme Activators and Inhibitors; |
| 应用: | URB602 is a selective inhibitor of MGL, exhibiting an IC50 of 28 µM for the rat brain enzyme. It does not inhibit fatty acid amide hydrolase (FAAH) at concentrations up to 100 µM, or other lipid metabolizing enzymes such as diacylglycerol lipase or cyclooxygenase-2.5 6 Inhibition of 2-AG hydrolysis is associated with enhanced stress-induced analgesia and may represent a novel drug target in pain and stress management. |
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