产品编号：E615300

产品规格：25mg

产品价格：面议

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产品详情

标准品编号:	E615300
名称:	ERK5-IN-1
别名:	11-Cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one;
CAS号:	1435488-37-1
分子式:	C₃₈H₄₆N₈O₃
分子量:	638.8
种类:	Research Tools; Molecular Biology; Enzyme Activators and Inhibitors;
应用:	ERK5-IN-1 is a potent selective ERK5 inhibitor, inhibiting EGFR-induced ERK5 autophosphorylation and ERK5 enzymatic activity. Orally bioavailable.
参考文献	Deng, X. et al. Eur. J. med. Chem., 70, 758 (2013); Elkins, J. et al.: J. Med. Chem., 56, 4413 (2013);