Dynarrestin

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产品编号:D826550

产品规格:50mg

产品价格:面议


产品详情

标准品编号: D826550
名称: Dynarrestin
别名: Ethyl-4-(4-(diethylamino)phenyl)-2-((2,4-difluorophenyl)amino)thiazole-5-carboxylate
CAS号: 2222768-84-3
分子式: C₂₂H₂₃F₂N₃O₂S
分子量: 431.5
种类: Standards; Enzyme Activators and Inhibitors;
应用: Dynarrestin is an dynein inhibitor. Inhibits hedgehog signaling in vitro (IC50 = 0.22 μM). Exhibits reversible inhibition of cytoplasmic dynein 1-dependent microtubule binding and cytoplasmic dynein 2-dependent intraflagellar transport. Inhibits tumor cell proliferation in a mouse medulloblastoma model.
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