产品编号：C375140

产品规格：10mg

产品价格：面议

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产品详情

标准品编号:	C375140
名称:	(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide
别名:	(S)-4-(4-Chlorophenyl)-N-(4-hydroxyphenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide; OTX015
CAS号:	202590-98-5
分子式:	C₂₅H₂₂ClN₅O₂S
分子量:	491.99
类别:	Research Tools;
应用:	(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide is an orally bioavailable, inhibitor of BRD2, BRD3, and BRD4 to AcH4 and shows anti-tumor activity in vitro and in vivo tumor models.
参考文献	Noel, J.K., et. al.: Mol. Cancer Ther. 12, 244 (2013)