BMS 182874 Hydrochloride

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产品编号:B695565

产品规格:2.5mg

产品价格:面议


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标准品编号: B695565
名称: BMS 182874 Hydrochloride
别名: 5-(Dimethylamino)-N-(3,4-dimethyl-5-isoxazolyl)-1-naphthalenesulfonamide hydrochloride
CAS号: 1215703-04-0
参考CAS: Free base: 153042-42-3
分子式: C₁₇H₁₉N₃O₃S • HCl
分子量: 345.403646
类别: Standards; Pharmaceutical/API Drug Impurities/Metabolites;
应用: BMS 182874 Hydrochloride, is a potent, selective, and competitive non-peptide endothelin ETAR antagonist (Ki = 48 nM). ET-A receptors are predominantly detected in peripheral tissues, especially in vascular smooth muscle tissues where they mediate vasoconstriction.
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