产品编号:B448535
产品规格:2.5mg
产品价格:面议
| 标准品编号: | B448535 |
| 名称: | Bisindolylmaleimide II |
| 别名: | 3-(1H-Indol-3-yl)-4-[1-[2-(1-methyl-2-pyrrolidinyl)ethyl]-1H-indol-3-yl]-1H-pyrrole-2,5-dione |
| CAS号: | 137592-45-1 |
| 分子式: | C₂₇H₂₆N₄O₂ |
| 分子量: | 438.52 |
| 类别: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | Bisindolylmaleimide II, is a potent ATP-competitive protein kinase C (PKC) inhibitor. In addition it inhibits PDK1 (IC50 = 14 μM), an important kinase in the insulin signaling pathway, and PKA (IC50 = 2.94 μM). |
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