BIIE 0246

我要购买

产品编号:B384503

产品规格:

产品价格:面议


产品详情

标准品编号: B384503
名称: BIIE 0246
别名: N-[(1S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide; AR-H 053591
CAS号: 246146-55-4
分子式: C₄₉H₅₇N₁₁O₆
分子量: 896.06
类别: Standards; Pharmaceutical/API Drug Impurities/Metabolites;
应用: BIIE 0246, is a selective non-peptide antagonist which binds to the neuropeptide NPY2-R in a competitive manner. Studies have also shown that BIIE 0246 is highly lipophilic and as a result BIIE 0246 builds up at membranes near the receptors.
文献