产品编号：B127623
产品规格：5mg
产品价格：面议
| 标准品编号: | B127623 |
| 名称: | BAZ2-ICR |
| 别名: | 4-[4-(1-Methyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]benzonitrile; |
| CAS号: | 1665195-94-7 |
| 分子式: | C₂₀H₁₉N₇ |
| 分子量: | 357.41 |
| 类别: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | BAZ2-ICR is a selective BAZ2 bromodomain inhibitor (IC50 values are 130 and 180 nM for BAZ2A and BAZ2B respectively). Exhibits 15-fold selectivity for the BAZ2 bromodomain over the CERC2 bromodomain and >100-fold selectivity over a range of other bromodomains. Accelerates FRAP recovery in a BAZ2A FRAP assay. |
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